Nitrendipine

Nitrendipine__L-type Ca channel blocker Dorsomorphin (dihydrochloride)

Product Name Nitrendipine
Description

L-type Ca channel blocker

Purity >98%
CAS No. 39562-70-4
Molecular Formula C18H20N2O6
Molecular Weight 360.37
Storage Temperature -20ºC
Shipping Temperature Shipped Ambient
Product Type Inhibitor
Solubility Soluble to 25 mM in ethanol and to 50 mM in DMSO
Source Synthetic
Appearance Yellow Crystalline Solid
SMILES CCOC(=O)C1=C(NC(=C(C1C2=CC(=CC=C2)N+(=O)O-)C(=O)OC)C)C
InChI InChI=1S/C18H20N2O6/c1-5-26-18(22)15-11(3)19-10(2)14(17(21)25-4)16(15)12-7-6-8-13(9-12)20(23)24/h6-9,16,19H,5H2,1-4H3
InChIKey PVHUJELLJLJGLN-UHFFFAOYSA-N
Safety Phrases Classification: Caution: Substance not fully tested yet.
Safety Phrases:
S22 – Do not breathe dust
S36/37/39 – Wear suitable protective clothing, gloves and eye/face protection
S24/25- Avoid contact with shin and eyes
Risk Phrases:
R62 – Possible risk of impaired fertility
Hazard Phrases:
H312-H332
Precautionary Phrases:
P280
Cite This Product Nitrendipine (StressMarq Biosciences Inc., Victoria BC CANADA, Catalog # SIH-320)
Alternative Names Ethyl methyl 2,6-dimethyl-4-(3-nitrophenyl)-1,4-dihydro-3,5-pyridinedicarboxylate
Research Areas Calcium Channels, Ion Channels, Neuroscience, Voltage-Gated Calcium Channels
PubChem ID 11931106
Scientific Background Nitrendipine is a dihydropyridine calcium channel blocker. It does so by binding effectively with the L-type calcium channels in smooth muscles thereby inactivating it and reducing the influx of calcium.
References 1.  Peterson B.Z., Tanada T.N., Catterall W.A. (1996) J Biol Chem. 271: 5293-5296.